• Acridinone-based anion transporters 

      McNaughton, Daniel A.; Macreadie, Lauren K.; Gale, Philip A.
      Published 2021
      The arrangement of hydrogen bond donors around a central lipophilic scaffold has proven a successful strategy in the development of potent chloride transporters. In this work, we revisit an acridinone 1,9-bis(thio)urea ...
      Open Access
      Article
    • Halide-selective, proton-coupled anion transport by phenylthiosemicarbazones 

      Howe, Ethan N.W.; Chang, Vai-Vai Tiffany; Wu, Xin; Fares, Mohamed; Lewis, William; Macreadie, Lauren K.; Gale, Philip A.
      Published 2022
      Phenylthiosemicarbazones (PTSCs) are proton-coupled anion transporters with pH-switchable behaviour known to be regulated by an imine protonation equilibrium. Previously, chloride/nitrate exchange by PTSCs was found to be ...
      Open Access
      Article
    • Synthesis, X-ray crystallographic analysis, DFT studies and biological evaluation of triazolopyrimidines and 2-anilinopyrimidines 

      Fares, Mohamed; Canfield, Peter; Alsherbiny, Muhammad A.; Lewis, William; Willis, Anthony C.; Li, Chun Guang; Neyts, Johan; Jochmans, Dirk; Gale, Philip A.; Keller, Paul A.
      Published 2022
      Inspired by the reported antiviral activity of pyrimidines and triazolopyrimidines, two series of 2-anilinopyrimidines (5a-e) and 1-aryl-[1,2,4]triazolo[4,3-a]pyrimidines (14a-k) were designed and synthesized as potential ...
      Open Access
      Article
    • Measuring anion transport selectivity: a cautionary tale 

      Wu, Xin; Gale, Philip A.
      Published 2021
      pH-dependent liposomal assays are often used to determine anion selectivity in transmembrane anion transport experiments. We discuss the validity and limitations of these assays, and provide guidelines for their use to ...
      Open Access
      Article
    • A Two-Dimensional Metallacycle Cross-Linked Switchable Polymer for Fast and Highly Efficient Phosphorylated Peptide Enrichment 

      Chen, Li-Jun; Humphrey, Sean; Zhu, Jun-Long; Zhu, Fan-Fan; Wang, Xu-Qing; Wang, Xiang; Wen, Jin; Yang, Hai-Bo; Gale, Philip A.
      Published 2021
      The selective and efficient capture of phosphopeptides is critical for comprehensive and in-depth phosphoproteome analysis. Reported here is a new switchable two-dimensional (2D) supramolecular polymer that can serve as ...
      Open Access
      Article