• Histone Deacetylase 2 (HDAC2) Inhibitors Containing Boron 

      Kavianpour, Poya; Gemmell, Madeleine C. M.; Kahlert, Jan U.; Rendina, Louis M.
      Published 2020
      Histone deacetylase enzymes (HDACs) are responsible for the global silencing of tumour‐suppressor genes. Treatment with a histone deacetylase inhibitor (HDACi) can reverse this process and restore normal cell function. ...
      Open Access
      Article
    • Gadolinium theranostics for the diagnosis and treatment of cancer 

      Robertson, Amy G.; Rendina, Louis M.
      Published 2021
      According to the World Health Organization (WHO), there were 18.1 million new cancer cases and 9.6 million cancer deaths reported worldwide in 2018. These numbers are expected to rise over the next decade, and the ...
      Open Access
      Article
    • Synthesis and tumour cell uptake studies of gadolinium(III)–phosphonium complexes 

      Hall, Andrew J.; Robertson, Amy G.; Hill, Leila R.; Rendina, Louis M.
      Published 2021
      The synthesis of a new series of Gd(III)-arylphosphonium complexes is described and the solution stability of selected compounds is reported. Their lipophilicity and uptake in human glial (SVG p12) and human glioblastoma ...
      Open Access
      Article
    • Fluoride binding by an anionic receptor: tuning the acidity of amide NH groups for basic anion hydrogen bonding and recognition 

      Montis, Ricardo; Bencini, Andrea; Coles, Simon J.; Conti, Luca; Fusaro, Luca; Gale, Philip A.; Giorgi, Claudia; Horton, Peter N.; Lippolis, Vito; Mapp, Lucy K.; Caltagirone, Claudia
      Published 2019
      Here we report a family of bis-amide receptors for anion binding that contain carboxylic acid groups vicinal to the amide function. Deprotonation of the carboxylic acids decreases the acidity of amide NHs, switching on ...
      Open Access
      Article
    • Supramolecular transmembrane anion transport: new assays and insights 

      Wu, Xin; Howe, Ethan N.W.; Gale, Philip A.
      Published 2018
      Transmembrane anion transport has been the focus of a number of supramolecular chemistry research groups for a number of years. Much of this research is driven by the biological relevance of anion transport and the search ...
      Open Access
      Article